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Dette derivatet kan acetyleres, hydroksyleres og glukuronideres. Cytokrom P-450 inkludert CYP3A kan spille en viktig rolle i reduksjon og oksidasjon av klonazepam. Eliminasjonshalveringstiden for klonazepam er vanligvis thirty til forty timer. Farmakokinetikken til klonazepam er doseuavhengig i hele doseringsområdet. Det er ingen bevis for at klon

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